About 18 results found for searched term "CGRP Receptor" (0.13 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2133 | MK-3207 hydrochloride | CGRP Receptor |
| MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM. | ||
| M3618 | MK-0974 | CGRP Receptor |
| Telcagepant | ||
| MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively. | ||
| M6504 | Olcegepant (BIBN-4096) | CGRP Receptor |
| BIBN-4096; BIBN 4096BS | ||
| Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. | ||
| M8322 | SB-268262 | CGRP Receptor |
| SB-268262 is a selective non-peptide antagonist at the CGRP1 receptor. | ||
| M10372 | Vazegepant hydrochloride | CGRP Receptor |
| Zavegepant, BHV-3500 hydrochloride | ||
| Vazegepant (BHV-3500) hydrochloride is a first-in-class, high affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM). Vazegepant hydrochloride may be useful in the effective treatment of lung inflammation associated with COVID-19. | ||
| M13931 | Calcitonin Gene Related Peptide (CGRP) (83-119), rat TFA | CGRP Receptor |
| Calcitonin Gene Related Peptide (CGRP) (83-119), rat (TFA) is a 37 amino acid calcitonin family of neuropeptide, acts through calcitonin receptor-like receptor (CRLR). | ||
| M13932 | HCGRP-(8-37) | CGRP Receptor |
| Human α-CGRP (8-37) | ||
| HCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor. | ||
| M13933 | MK-3207 | CGRP Receptor |
| MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. | ||
| M13934 | Olcegepant hydrochloride | CGRP Receptor |
| BIBN-4096 hydrochloride; BIBN4096BS hydrochloride | ||
| Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. | ||
| M13935 | Rat CGRP-(8-37) | CGRP Receptor |
| Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist. | ||
| M24721 | Erenumab | CGRP Receptor |
| Erenumab is a fully human monoclonal antibody. Erenumab inhibits the calcitonin gene–related peptide (CGRP) receptor. Erenumab can be used for the prevention of episodic migraine. | ||
| M24771 | Eptinezumab | CGRP Receptor |
| Eptinezumab is a human monoclonal antibody. Eptinezumab binds to calcitonin gene-related peptide (CGRP) and blocks its binding to the receptor. Eptinezumab can be used for the prevention of migraine in adults. | ||
| M28198 | Vazegepant | CGRP Receptor |
| Zavegepant; BHV-3500 | ||
| Vazegepant (Zavegepant) is a first-in-class CGRP receptor antagonist with potential for acute studies in migraine. | ||
| M50213 | CGRP antagonist 1 | CGRP Receptor |
| CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki and IC50 values of 1.7 nM and 5.7 nM, respectively. | ||
| M50214 | AC 187 TFA | Amyloid |
| AC 187 TFA is a potent, orally active and neuroprotective amylin receptor antagonist with an IC50 of 0.48 nM and a Ki of 0.275 nM. AC 187 TFA is more selective for amylin receptors than calcitonin and CGRP receptors. | ||
| M53227 | [Tyr22] Calcitonin Gene Related Peptide, (22-37), rat | CGRP Receptor |
| [Tyr22] Calcitonin Gene Related Peptide, (22-37), rat is a fragments 22-37 of rat calcitonin gene related peptide (CGRP), targeting CGRP receptor and adenylate cyclase. | ||
| M53230 | Calcitonin Gene Related Peptide (CGRP) II, rat | CGRP Receptor |
| Calcitonin Gene Related Peptide (CGRP) II, rat, a CGRP receptor activator, is a potent and long-lasting vasodilator. | ||
| M53900 | Adrenomedullin (AM) (22-52), human | CGRP Receptor |
| Adrenomedullin (AM) (22-52), human is an adrenomedullin receptor antagonist, and also antagonizes the calcitonin generelated peptide (CGRP) receptor in the hindlimb vascular bed of the cat. | ||
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